Lebelo, M.T. (Maphuti); Joubert, Anna Margaretha; Visagie, M.H. (Michelle Helen)
(MDPI, 2020-09)
2-Methoxyestradiol (2ME), a 17β-estradiol metabolite, exerts anticancer properties
in vitro and in vivo. To address 2ME’s low bioavailability, research led to the in silico design
of sulphamoylated 2ME analogues. However, ...