Repsold, Lisa; Pretorius, Etheresia; Joubert, Annie M.
(BioMed Central, 2014-06-07)
BACKGROUND: 2-Methoxyestradiol is known to have antitumour and antiproliferative action in vitro and in vivo.
However, when 2-methoxyestradiol is orally administered, it is rapidly oxidized by the enzyme 17β-hydroxyster ...