Helena, Jolene Michelle; Joubert, Anna Margaretha; Mabeta, Peaceful Lucy; Coetzee, Magdalena; Lakier, Roy; Mercier, Anne Elisabeth
(MDPI, 2021-08-17)
2-Ethyl-3-O-sulfamoyl-estra-1,3,5(10)16-tetraene (ESE-16) is an in silico-designed estradiol
analogue which has improved the parent compound’s efficacy in anti-cancer studies. In this proofof-
concept study, the potential ...