Structure−activity relationship studies reveal new astemizole analogues active against Plasmodium falciparum in vitro

dc.contributor.authorMambwe, Dickson
dc.contributor.authorKumar, Malkeet
dc.contributor.authorFerger, Richard
dc.contributor.authorTaylor, Dale
dc.contributor.authorNjoroge, Mathew
dc.contributor.authorCoertzen, Dina
dc.contributor.authorReader, Janette
dc.contributor.authorVan der Watt, Mariette Elizabeth
dc.contributor.authorBirkholtz, Lyn-Marie
dc.contributor.authorChibale, Kelly
dc.date.accessioned2021-10-15T11:57:00Z
dc.date.issued2021-08
dc.description.abstractPlease read abstract in the article.en_ZA
dc.description.departmentBiochemistryen_ZA
dc.description.departmentGeneticsen_ZA
dc.description.departmentMicrobiology and Plant Pathologyen_ZA
dc.description.embargo2022-08-02
dc.description.librarianhj2021en_ZA
dc.description.urihttps://pubs.acs.org/journal/aidcbcen_ZA
dc.identifier.citationMambwe, D., Kumar, M., Ferger, R. et al. 2021, 'Structure−activity relationship studies reveal new astemizole analogues active against Plasmodium falciparum in vitro', ACS Medicinal Chemistry Letters, vol. 12, no. 8, pp. 1333-1341.en_ZA
dc.identifier.issn1948-5875
dc.identifier.other10.1021/acsmedchemlett.1c00328
dc.identifier.urihttp://hdl.handle.net/2263/82130
dc.language.isoenen_ZA
dc.publisherAmerican Chemical Societyen_ZA
dc.rights© 2021 American Chemical Societyen_ZA
dc.subjectAstemizoleen_ZA
dc.subjectPlasmodium falciparumen_ZA
dc.subjectRepositioningen_ZA
dc.subjectHuman ether-a-go-go-related geneen_ZA
dc.titleStructure−activity relationship studies reveal new astemizole analogues active against Plasmodium falciparum in vitroen_ZA
dc.typePostprint Articleen_ZA

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